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2027年考研必胜卡--药学综合第42天!

  • 2026-02-02 20:50:46
2027年考研必胜卡--药学综合第42天!

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考研

2024

2024

加油

1

为了增加甲硝唑溶解度,使用水-乙醇混合溶剂作为( )

A.潜溶剂

B.助悬剂

C.防腐剂

D.助溶剂

E.增溶剂

2

脂溶性药物依靠药物分子在膜两侧的浓度差,从膜的高浓度一侧向低浓度转运药物的方式是( )

A、膜动转运

B、简单扩散

C、主动转运

D、滤过

E、易化扩散

答案与解析

1.第一题答案:C

该题出自及解析:

本题考查液体制剂常用附加剂。液体制剂常用附加剂有:

(1)增溶剂:增溶是指难溶性药物在表面活性剂的作用下,在溶剂中增加溶解度并形成溶液的过程。常用增溶剂为聚山梨酯类、 聚氧乙烯脂肪酸酯类等;

(2) 助溶剂:难溶性药物与加入的第三种物质在溶剂中形成可溶性分子间的络合物、缔合物或复盐等,以增加药物在溶剂中的溶解度。助溶剂多为某些有机酸及其盐类如苯甲酸、碘化钾等;

(3) 潜溶剂:系指能形成氢键以增加难溶性药物溶解度的混合溶剂,能与水形成潜溶剂的有乙醇、丙二醇、甘油、聚乙二醇等;

(4)防腐剂:又称抑菌剂,系指具有抑菌作用,能抑制微生物生长繁殖的物质。常用的防腐剂有苯甲酸与苯甲酸钠、对羟基苯甲酸酯类、山梨酸与山梨酸钾、苯扎溴铵等。其他附加剂有矫味剂、着色剂等。助悬剂是指能增加混悬剂中分散介质的黏度,降低药物微粒的沉降速度或增加微粒亲水性的附加剂,包括低分子助悬剂如甘油,高分子助悬剂如果胶、甲基纤维素,硅皂土和触变胶等。

2.第二题答案:B

该题出自及解析:

本题考查药物的转运方式。药物的转运方式有被动转运、载体转运和膜动转运。被动转运是物质从高浓度区域向低浓度区域的转运,转运速度与膜两侧的浓度差成正比,转运过程不需要载体,不消耗能量。被动转运包括滤过(水溶性小分子物质)和简单扩散(脂溶性药物)。载体转运由载体介导,生物膜中的蛋白质具有载体的作用。载体转运有主动转运和易化扩散两种方式。药物通过生物膜转运时,借助载体或酶促系统,可以从膜的低浓度一侧向高浓度一侧转运,这种过程称为主动转运;易化扩散又称中介转运,是指一些物质在细胞膜载体的帮助下,由膜的高浓度一侧向低浓度一侧转运的过程,与主动转运不同之处在于:易化扩散不消耗能量,而且是顺浓度梯度转运。生物膜具有一定的流动性,它可以通过主动变形,膜凹陷吞没液滴或微粒,将某些物质摄入细胞内或从细胞内释放到细胞外,此过程称膜动转运。

答案参考书目:

药理学:第八版,《人民卫生出版社》,朱依淳主编(黑字体);第七版,《人民卫生出版社》,杨宝峰主编(红字体)

药物化学:第二版,《化学工业出版社》,尤启冬主编(黑字体);第八版,《人民卫生出版社》,尤启冬主编(红字体)

目前参考书目:第一版,《科学出版社》,鄢明,成志毅主编

药剂学:第七版,《人民卫生出版社》,崔福德主编(黑字体);第八版,《人民卫生出版社》,方亮主编(红字体)

药物分析:第七版,《人民卫生出版社》,杭太俊主编(黑字体);第八版,《人民卫生出版社》,杭太俊主编(红字体)

每日两个知识点:

恭喜你!当你看到这里的时候,你成功打卡42天!

离成功又近了一步!

离2027考研还有322天!

加油!

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  1. CONNECT:[ UseTime:0.000503s ] mysql:host=127.0.0.1;port=3306;dbname=b_mffb;charset=utf8mb4
  2. SHOW FULL COLUMNS FROM `fenlei` [ RunTime:0.000735s ]
  3. SELECT * FROM `fenlei` WHERE `fid` = 0 [ RunTime:0.000293s ]
  4. SELECT * FROM `fenlei` WHERE `fid` = 63 [ RunTime:0.000259s ]
  5. SHOW FULL COLUMNS FROM `set` [ RunTime:0.000585s ]
  6. SELECT * FROM `set` [ RunTime:0.000201s ]
  7. SHOW FULL COLUMNS FROM `article` [ RunTime:0.000504s ]
  8. SELECT * FROM `article` WHERE `id` = 475316 LIMIT 1 [ RunTime:0.000539s ]
  9. UPDATE `article` SET `lasttime` = 1770294510 WHERE `id` = 475316 [ RunTime:0.004593s ]
  10. SELECT * FROM `fenlei` WHERE `id` = 66 LIMIT 1 [ RunTime:0.000237s ]
  11. SELECT * FROM `article` WHERE `id` < 475316 ORDER BY `id` DESC LIMIT 1 [ RunTime:0.006399s ]
  12. SELECT * FROM `article` WHERE `id` > 475316 ORDER BY `id` ASC LIMIT 1 [ RunTime:0.001640s ]
  13. SELECT * FROM `article` WHERE `id` < 475316 ORDER BY `id` DESC LIMIT 10 [ RunTime:0.009550s ]
  14. SELECT * FROM `article` WHERE `id` < 475316 ORDER BY `id` DESC LIMIT 10,10 [ RunTime:0.001604s ]
  15. SELECT * FROM `article` WHERE `id` < 475316 ORDER BY `id` DESC LIMIT 20,10 [ RunTime:0.002404s ]
0.101400s